A-485

Vendor: Abmole

Type: Molecular

SKU: M9561

$368.00 USD
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Documents

Coa

Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
A-485 is a potent and selective HAT inhibitor of p300/CBP in vitro with an IC50 of 10 nM in a p300 TR-FRET assay and 3 nM in a CBP TR-FRET assay with selectivity > 1000-fold over closely related HATs.
Casnumber
1889279-16-6
Formula
C25H24F4N4O5
Mw
536.48
Psmiles
CNC(=O)NC1=CC=C2C(=C1)CCC23OC(=O)N(CC(=O)N(CC4=CC=C(F)C=C4)C(C)C(F)(F)F)C3=O
Purity
>99%
Solubility
DMSO ≥ 60 mg/mL
A-485

A-485

$368.00 USD