A1874

Vendor: Abmole

Type: Molecular

SKU: M9396

$759.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
A1874 is a BRD4-degrading PROTAC which inhibits many cancer cell lines proliferation, with DC50 of 32 nM (induce BRD4 degradation in cells).
Casnumber
2064292-12-0
Formula
C58H62Cl3F2N9O7S
Mw
1173.59
Psmiles
COC1=C(NC(=O)C2NC(CC(C)(C)C)C(C#N)(C2C3=C(F)C(=CC=C3)Cl)C4=C(F)C=C(Cl)C=C4)C=CC(=C1)C(=O)NCCOCCOCCOCCNC(=O)CC5N=C(C6=CC=C(Cl)C=C6)C7=C(SC(=C7C)C)[N]8C(=NN=C58)C
Purity
>99.0%
Solubility
DMSO ≥ 60 mg/mL
A1874

A1874

$759.00 USD