Alvimopan dihydrate

Vendor: Abmole

Type: Molecular

SKU: M5403

$184.00 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively).
Casnumber
170098-38-1
Formula
C25H36N2O6
Mw
460.56
Psmiles
O.O.CC1CN(CCC1(C)C2=CC=CC(=C2)O)CC(CC3=CC=CC=C3)C(=O)NCC(O)=O
Purity
>98.5%
Solubility
DMSO 30 mg/mL
Target synonyms
LY 246736 dihydrate; ADL 8-2698 dihydrate
Alvimopan dihydrate

Alvimopan dihydrate

$184.00 USD