API-1

Vendor: Abmole

Type: Molecular

SKU: M9571

$304.75 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
API-1 is a Pin1 inhibitor with an IC50 of 72.3 nM. API-1 directly and specifically binds to the Pin1 peptidyl-prolyl isomerase (PPIase) domain and potently inhibits Pin1 cis-trans isomerizing activity.
Casnumber
680622-70-2
Formula
C15H13F3N6O2
Mw
366.30
Psmiles
NC1=NC2=NC=NC2=C([NH]1)OCC3=CC=C(CNC(=O)C(F)(F)F)C=C3
Purity
>98%
Solubility
DMSO ≥ 100 mg/mL
API-1

API-1

$304.75 USD