Aprocitentan

Vendor: Abmole

Type: Molecular

SKU: M13956

$189.75 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively.
Casnumber
1103522-45-7
Formula
C16H14Br2N6O4S
Mw
546.19
Psmiles
C1=CC(=CC=C1C2=C(N=CN=C2OCCOC3=NC=C(C=N3)Br)NS(=O)(=O)N)Br
Purity
99.77%
Solubility
DMSO 23 mg/mL
Target synonyms
ACT-132577
Aprocitentan

Aprocitentan

$189.75 USD