ARP-100

Vendor: Abmole

Type: Molecular

SKU: M30518

$113.85 USD
Shipping calculated at checkout.

Documents

Coa

Available in stock (500)

  • Customs clearance fees may apply
  • Worldwide shipping available.
For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
ARP-100 is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM). ARP-100 interacts with S1＇ pocket of MMP-2 and shows anti-invasive properties in an in vitro model of invasion on matrigel. ARP-100 shows the less inhibitory activity towards MMP-1 (>50 μM), MMP-3 (4.5 μM), MMP-7 (>50 μM), and MMP-9 (0.2 μM).
Casnumber
704888-90-4
Formula
C17H20N2O5S
Mw
364.42
Psmiles
CC(C)ON(CC(=O)NO)[S](=O)(=O)C1=CC=C(C=C1)C2=CC=CC=C2
Purity
≥99.0%
Solubility
DMSO 100 mg/mL (ultrasonic)
ARP-100

ARP-100

$113.85 USD