ARQ-087

Vendor: Abmole

Type: Molecular

SKU: M6158

$276.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
ARQ 087 is a novel, ATP competitive, small molecule, multi-kinase inhibitor with potent in vitro and in vivo activity against FGFR addicted cell lines and tumors. ARQ 087 exhibited IC50 values of 1.8 nM for FGFR2, and 4.5 nM for FGFR1 and 3.
Casnumber
1234356-69-4
Formula
C29H29FN4O
Mw
468.57
Psmiles
COCCNCCC1=CC(=CC=C1)NC2=NC3=C(CC(C4=CC=CC=C4F)C5=C3C=CC=C5)C=N2
Purity
>99%
Solubility
DMSO 84 mg/mL
Target synonyms
Derazantinib
ARQ-087

ARQ-087

$276.00 USD