ARV-766

Vendor: Abmole

Type: Molecular

SKU: M25607

$1,150.00 USD
Shipping calculated at checkout.

Documents

Coa

Available in stock (500)

  • Customs clearance fees may apply
  • Worldwide shipping available.
For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
ARV-766 is an orally active and potent proteolysis targeting chimera (PROTAC) protein degrader. ARV-766 degrades wild-type androgen receptor (AR) but also relevant AR LBD mutants, including the most prevalent AR L702H, H875Y, and T878A mutations. ARV-766 has the potential to be first- and best-in class PROTAC AR degrader in mCRPC.
Casnumber
2750830-09-0
Formula
C45H54FN7O6
Mw
807.95
Psmiles
COC1=C(C=CC(=C1)OC2C(C)(C)C(NC(=O)C3=CC=C(C=C3)N4CCC(CC4)CN5CCN(CC5)C6=CC(=C(C=C6)C(=O)NC7CCC(=O)NC7=O)F)C2(C)C)C#N
Purity
>99.0%
Solubility
DMSO 90 mg/mL
Target synonyms
Luxdegalutamide
ARV-766

ARV-766

$1,150.00 USD