AZ194

Vendor: Abmole

Type: Molecular

SKU: M29408

$333.50 USD
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Coa

Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
AZ194 is a first-in-class, orally active inhibitor of CRMP2-Ubc9 interaction and inhibitor of NaV1.7 (IC50=1.2 μM). AZ194 blocks SUMOylation of CRMP2 to selectively reduce the amount of surface-expressed NaV1.7. Antinociceptive effects.
Casnumber
2241651-99-8
Formula
C34H31F2N3O3
Mw
567.63
Psmiles
COC1=C(C=CC(=C1)C(=O)N2CCC(CC2)C3=NC4=CC=CC=C4N3CC5=CC(=CC=C5)F)OCC6=CC(=CC=C6)F
Purity
≥99.0%
Solubility
DMSO 30 mg/mL (ultrasonic)
AZ194

AZ194

$333.50 USD