BMS-536924

Vendor: Abmole

Type: Molecular

SKU: M1957

$166.75 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Bms-536924 is an orally active, competitive and selective insulin-like growth factor receptor (IGF-1R) kinase and insulin receptor (IR) inhibitor with IC50 of 100 nM and 73 nM, respectively. It also showed moderate inhibitory activity against Mek, Fak and Lck, but almost no inhibitory activity against Akt1 and MAPK1/2.
Casnumber
468740-43-4
Formula
C25H26ClN5O3
Mw
479.96
Psmiles
CC1=C2N=C([NH]C2=CC(=C1)N3CCOCC3)C4=C(NCC(O)C5=CC=CC(=C5)Cl)C=CNC4=O
Purity
>99.0%
Solubility
DMSO 66 mg/mL
BMS-536924

BMS-536924

$166.75 USD