BRD4770

Vendor: Abmole

Type: Molecular

SKU: M8397

$109.25 USD
Shipping calculated at checkout.

Documents

Coa

Available in stock (500)

  • Customs clearance fees may apply
  • Worldwide shipping available.
For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
BRD4770 is a histone methyltransferase G9a inhibitor. BRD4770 inhibited the dimethylation and trimethylation of H3K9, EC50 was 5 µM, and had little effect on H3K27me3, H3K36me3, H3K4me3, and H3K79me3. BRD4770 activates the ataxic telangiectasia mutation (ATM) pathway and induces cell senescence.
Casnumber
1374601-40-7
Formula
C25H23N3O3
Mw
413.47
Psmiles
COC(=O)C1=CC=C2[N](CCCC3=CC=CC=C3)C(=NC2=C1)NC(=O)C4=CC=CC=C4
Purity
>99.0%
Solubility
DMSO: 5 mg/mL (warmed)
BRD4770

BRD4770

$109.25 USD