CHR-6494 TFA

Vendor: Abmole

Type: Molecular

SKU: M59246

$230.00 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
CHR-6494 TFA is a potent and selective inhibitor of haspin, with an IC50 of 2 nM. CHR-6494 TFA induces cell cycle arrest at G2/M, inhibits cell proliferation, and promotes apoptosis in multiple cancer cell lines. CHR-6494 TFA inhibits histone H3T3 phosphorylation.
Casnumber
1458630-17-5
Formula
C18H17F3N6O2
Mw
406.36
Psmiles
CCCNC1=NN2C(=NC=C2C3=CC4=C(C=C3)NN=C4)C=C1.C(=O)(C(F)(F)F)O
Purity
≥98.0%
Solubility
DMSO 40 mg/mL
Target synonyms
CHR 6494 trifluoroacetate
CHR-6494 TFA

CHR-6494 TFA

$230.00 USD