Clobenpropit dihydrobromide

Vendor: Abmole

Type: Molecular

SKU: M28480

$207.00 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Clobenpropit dihydrobromide is a potent histamine H3R antagonist/inverse agonist with a pEC50 of 8.07 for histamine H3LR. Clobenpropit dihydrobromide acts as partial agonist at histamine H4 receptors (Ki 13 nM). Clobenpropit dihydrobromide also binds to serotonin 5-HT3 receptors (Ki 7.4 nM) and α2A/α2C adrenoceptors (Ki 17.4/7.8 nM). Clobenpropit dihydrobromide increases apoptosis.
Casnumber
145231-35-2
Formula
C14H19Br2ClN4S
Mw
470.65
Psmiles
C1=CC(=CC=C1CN=C(N)SCCCC2=CN=CN2)Cl.Br.Br
Purity
≥99.0%
Solubility
DMSO 100 mg/mL (ultrasonic)
Clobenpropit dihydrobromide

Clobenpropit dihydrobromide

$207.00 USD