Dalpiciclib

Vendor: Abmole

Type: Molecular

SKU: M10930

$805.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Dalpiciclib (SHR-6390) is a highly selective, oral bioavailable inhibitor of CDK4/6 that is used against CDK4 (IC50=12.4 nM) and CDK6 (IC50=9.9 nM) is equivalent. SHR6390 exerts potent antitumor activity in esophageal squamous cell carcinoma by inhibiting phosphorylated Rb protein and inducing G1 cell cycle blocking.
Casnumber
1637781-04-4
Formula
C25H30N6O2
Mw
446.54
Psmiles
CC1=C(C(=O)N(C2=NC(=NC=C12)NC3=NC=C(C=C3)C4CCNCC4)C5CCCC5)C(=O)C
Purity
100.0%
Target synonyms
SHR-6390
Dalpiciclib

Dalpiciclib

$805.00 USD