dBET1

Vendor: Abmole

Type: Molecular

SKU: M9237

$189.75 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
dBET1 is a potent BRD4 protein degrader with an EC50 of 430 nM. dBET1 is a PROTAC that composes of (+)-JQ1 linked to NSC 527179 with a linker.
Casnumber
1799711-21-9
Formula
C38H37ClN8O7S
Mw
785.27
Psmiles
CC1=C(C)C2=C(S1)[N]3C(=NN=C3C(CC(=O)NCCCCNC(=O)COC4=CC=CC5=C4C(=O)N(C6CCC(=O)NC6=O)C5=O)N=C2C7=CC=C(Cl)C=C7)C
Purity
≥99.0%
Solubility
DMSO 40 mg/mL
dBET1

dBET1

$189.75 USD