dBET57

Vendor: Abmole

Type: Molecular

SKU: M10380

$276.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
dBET57 is a novel BRD4 heterobifunctional small-molecule ligand (PROTAC) which exhibits significant and selective degradation of BRD4 BD1 but is inactive on BRD4 BD2.
Casnumber
1883863-52-2
Formula
C34H31ClN8O5S
Mw
699.18
Psmiles
CC1=C(C)C2=C(S1)[N]3C(=NN=C3C(CC(=O)NCCNC4=CC=CC5=C4C(=O)N(C6CCC(=O)NC6=O)C5=O)N=C2C7=CC=C(Cl)C=C7)C
Purity
>99%
Solubility
DMSO ≥ 100 mg/mL
Target synonyms
dBET-57
dBET57

dBET57

$276.00 USD