EED226

Vendor: Abmole

Type: Molecular

SKU: M5243

$552.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
EED226 is an effective, selective and orally active Polycomb reactive complex 2 (PRC2) inhibitor. When h3k27me0 peptide is used as substrate, ic50=23.4 nm; With mononucleosome as substrate, ic50=53.5 nm. It is a first in class, effective, orally bioavailable inhibitor of embryonic ectodermal development (EED) with strong anticancer effect.
Casnumber
2083627-02-3
Formula
C17H15N5O3S
Mw
369.40
Psmiles
C[S](=O)(=O)C1=CC=C(C=C1)C2=CN=C(NCC3=CC=CO3)[N]4C=NN=C24
Purity
>99.0%
Solubility
73 mg/mL in DMSO
EED226

EED226

$552.00 USD