Endoxifen (Z-isomer)

Vendor: Abmole

Type: Molecular

SKU: M27811

$287.50 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Endoxifen Z-isomer is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen inhibits hERG tail currents at 50 mV in a concentration-dependent manner with IC50 values of 1.6 μM.
Casnumber
112093-28-4
Formula
C25H27NO2
Mw
373.49
Psmiles
CCC(=C(C1=CC=C(C=C1)O)C2=CC=C(C=C2)OCCNC)C3=CC=CC=C3
Purity
≥99.0%
Solubility
DMSO 50 mg/mL (ultrasonic)
Endoxifen (Z-isomer)

Endoxifen (Z-isomer)

$287.50 USD