Ensifentrine

Vendor: Abmole

Type: Molecular

SKU: M11547

$230.00 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Ensifentrine (RPL-554) is an inhaled, pioneering dual inhibitor of phosphodiesterase 3 (PDE3) and PDE4 with IC50 of 0.4 nM and 1479 nM, respectively. Ensifentrine has bronchoprotective and anti-inflammatory activity and can be used to study chronic obstructive pulmonary disease (COPD).
Casnumber
1884461-72-6
Formula
C26H31N5O4
Mw
477.56
Psmiles
CC1=CC(=C(C(=C1)C)N=C2C=C3C4=CC(=C(C=C4CCN3C(=O)N2CCNC(=O)N)OC)OC)C
Purity
>99%
Solubility
DMSO ≥ 10 mg/mL
Target synonyms
RPL-554;Ensifentrinum, Ensifentrina
Ensifentrine

Ensifentrine

$230.00 USD