FM-381

Vendor: Abmole

Type: Molecular

SKU: M10698

$241.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
FM-381 is a potent, covalent, reversible JAK3 inhibitor that targets the Cys909 site. FM-381 for JAK3 IC50 The value is 127 pM, which is 410, 2700, and 3600 times more selective than JAK1, JAK2, and TYK2, respectively.
Casnumber
2226521-65-7
Formula
C24H24N6O2
Mw
428.49
Psmiles
CN(C)C(=O)/C(=C/C1=CC=C(O1)C2=NC3=CN=C4[NH]C=CC4=C3[N]2C5CCCCC5)C#N
Purity
>99.0%
Solubility
DMSO ≥ 10 mg/mL
FM-381

FM-381

$241.50 USD