Gartisertib

Vendor: Abmole

Type: Molecular

SKU: M11251

$736.00 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Gartisertib (VX-803) is an ATP-competitive, orally active, selective ATR inhibitor with Ki<150 pM. Gartisertib inhibits atR-driven phosphorylation of checkpoint kinase-1 (Chk1) with an IC50 value of 8 nM. It has antitumor activity.
Casnumber
1613191-99-3
Formula
C25H29F2N9O3
Mw
541.55
Psmiles
NC1=N[N]2C=C(F)C=NC2=C1C(=O)NC3=C(N4CCC(CC4)C(=O)N5CCN(CC5)C6COC6)C(=CN=C3)F
Purity
>99%
Solubility
DMSO ≥ 10 mg/mL
Target synonyms
VX-803; M4344; ATR inhibitor 2
Gartisertib

Gartisertib

$736.00 USD