GDC-0276

Vendor: Abmole

Type: Molecular

SKU: M28535

$851.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
GDC-0276 is a potent, selective, reversible and orally active NaV1.7 inhibitor with an IC50 value of 0.4 nM. GDC-0276 is well tolerated and exhibits a good pharmacokinetic profile. GDC-0276 has the potential for the treatment of pain and to address shortcomings of existing pain medications, such as addiction and off-target side effects.
Casnumber
1494581-70-2
Formula
C24H31FN2O4S
Mw
462.58
Psmiles
C1CN(C1)S(=O)(=O)NC(=O)C2=C(C=C(C(=C2)C3CC3)OCC45CC6CC(C4)CC(C6)C5)F
Purity
≥99.0%
Solubility
DMSO 100 mg/mL (ultrasonic)
GDC-0276

GDC-0276

$851.00 USD