GS-9876 (lanraplenib)

Vendor: Abmole

Type: Molecular

SKU: M20799

$1,150.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Lanraplenib (GS-9876, GS-SYK) is a potent, highly selective and orally active inhibitor of Spleen Tyrosine Kinase (SYK) with IC50 of 9.5 nM. Lanraplenib inhibits SYK activity in platelets via the glycoprotein VI (GPVI) receptor without prolonging bleeding time (BT) in monkeys or humans.
Casnumber
1800046-95-0
Formula
C23H25N9O
Mw
443.5
Psmiles
NC1=CN=CC(=N1)C2=C[N]3C=CN=C3C(=N2)NC4=CC=C(C=C4)N5CCN(CC5)C6COC6
Purity
>99%
Solubility
DMSO 89 mg/mL
Target synonyms
GS-SYK
GS-9876 (lanraplenib)

GS-9876 (lanraplenib)

$1,150.00 USD