GSK3368715 2HCl

Vendor: Abmole

Type: Molecular

SKU: M10637

$207.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
GSK3368715 2HCl is a novel potent, orally active, reversible type I protein arginine methyltransferases (PRMTs) inhibitor, with IC50 values of 3.1 nM, 48 nM, 1148 nM, 5.7 nM and 1.7 nM for PRMT1, PRMT3, PRMT4, PRMT6, PRMT8, respectively.
Casnumber
1628925-77-8
Formula
C20H40Cl2N4O2
Mw
439.46
Psmiles
CCOCC1(CCC(CC1)C2=C(C=NN2)CN(C)CCNC)COCC.Cl.Cl
Purity
>99%
Solubility
DMSO ≥ 100 mg/mL; Water ≥ 90 mg/mL
Target synonyms
EPZ019997 2HCl
GSK3368715 2HCl

GSK3368715 2HCl

$207.00 USD