GSK3987

Vendor: Abmole

Type: Molecular

SKU: M29748

$138.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
GSK3987 is a pan LXRα/β agonist with EC50s of 50 nM, 40 nM for LXRα-SRC1 and LXRβ-SRC1, respectively. GSK3987 increases the expression of ABCA1 and SREBP-1c. GSK3987 induces cellular cholesterol efflux and triglyceride accumulation.
Casnumber
264206-85-1
Formula
C24H20N2O3
Mw
384.43
Psmiles
COC1=CC=C(NC2=C(C(=O)N(CC3=CC=CC=C3)C2=O)C4=CC=CC=C4)C=C1
Purity
≥99.0%
Solubility
DMSO 100 mg/mL (ultrasonic)
GSK3987

GSK3987

$138.00 USD