GSK481

Vendor: Abmole

Type: Molecular

SKU: M5209

$155.25 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
GSK481 is a highly effective, selective and specific RIPK1 inhibitor with an IC50 value of 1.3 nM, which can inhibit the phosphorylation of Ser166 in wild-type human RIPK1 (IC50 value of 2.8 nM). The IC50 value of GSK481 against U937 cells was 10 nM.
Casnumber
1622849-58-4
Formula
C21H19N3O4
Mw
377.39
Psmiles
CN1C(=O)C(COC2=CC=CC=C12)NC(=O)C3=NOC(=C3)CC4=CC=CC=C4
Purity
99.90%
Solubility
DMSO 70 mg/mL
Target synonyms
GSK481
GSK481

GSK481

$155.25 USD