GSK620

Vendor: Abmole

Type: Molecular

SKU: M10760

$170.20 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
GSK620 is a potent orally active pan-BD2 inhibitor with good broad-spectrum selectivity, developability, and in vivo oral pharmacokinetics, and is highly selective against the BET-BD2 family protein, with a selectivity of more than 200 times that of all other BET bromodomains. GSK620 exhibits an anti-inflammatory phenotype in human whole blood.
Casnumber
2088410-46-0
Formula
C18H19N3O3
Mw
325.36
Psmiles
CNC(=O)C1=CC(=CN(CC2=CC=CC=C2)C1=O)C(=O)NC3CC3
Purity
>99.0%
Solubility
DMSO ≥ 60 mg/mL
GSK620

GSK620

$170.20 USD