GSK864

Vendor: Abmole

Type: Molecular

SKU: M8651

$379.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
GSK864 is a cell penetrant, potent and selective allosteric inhibitor of isocitrate dehydrogenase 1 (IDH1) that potently inhibits intracellular 2-hydroxyglutarate (2-HG) production in HT-1080 cells.
Casnumber
1816331-66-4
Formula
C30H31FN6O4
Mw
558.6
Psmiles
CC1=CC(=CC(=C1OC)C)NC(=O)C2=NN(C3=C2CN(CC3(C)C(=O)N)C(=O)C4=CC=CN4)CC5=CC=C(C=C5)F
Purity
99.99%
Solubility
DMSO: 10 mg/mL
GSK864

GSK864

$379.50 USD