HJC0197

Vendor: Abmole

Type: Molecular

SKU: M11263

$178.25 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
HJC0197 is a potent antagonist of Epac1 (the exchange protein directly activated by cAMP 1) and Epac2 (IC50=5.9 μM for Epac2). HJC0197 selectively blocked camp-induced Epac activation. HJC0197 inhibited epAC1-mediated RAP1-GDP exchange activity in the presence of isoconcentration of cAMP.
Casnumber
1383539-73-8
Formula
C19H21N3OS
Mw
339.45
Psmiles
CC1=CC(=C(C)C=C1)CSC2=NC(=C(C#N)C(=O)N2)C3CCCC3
Purity
>98%
Solubility
DMSO ≥ 40 mg/mL
HJC0197

HJC0197

$178.25 USD