Inobrodib

Vendor: Abmole

Type: Molecular

SKU: M21109

$368.00 USD
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Coa

Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Inobrodib (CCS1477, CBP-IN-1) is an orally active, potent and selective p300/CBP inhibitor. inobrodib binds to p300 and CBP with Kd values of 1.3 and 1.7 nM and has a 170/130 fold selectivity compared to BRD4 with a Kd of 222 nM. Inobrodib (CCS1477) acts by inhibiting the expression and function of androgen receptor (AR) and by inhibiting c-Myc.
Casnumber
2222941-37-7
Formula
C30H32F2N4O3
Mw
534.6
Psmiles
COC1CCC(CC1)[N]2C(=NC3=CC(=CC=C23)C4=C(C)ON=C4C)C5CCCC(=O)N5C6=CC(=C(F)C=C6)F
Purity
>99.0%
Solubility
DMSO 90 mg/mL
Target synonyms
CCS1477; CBP-IN-1; CBP/p300-IN-4
Inobrodib

Inobrodib

$368.00 USD