IRL 2500

Vendor: Abmole

Type: Molecular

SKU: M28815

$356.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
IRL 2500 is a potent Endothelin receptor antagonist. IRL 2500 shows IC50 values of 1.3 and 94 nM for ETB and ETA receptors, respectively. IRL 2500 inhibits ETB receptor-mediated blood pressure increase and renal vascular resistance in rats in vivo.
Casnumber
169545-27-1
Formula
C36H35N3O4
Mw
573.68
Psmiles
CC1=CC(=CC(=C1)C(=O)N(C)C(CC2=CC=C(C=C2)C3=CC=CC=C3)C(=O)NC(CC4=CNC5=CC=CC=C54)C(=O)O)C
Purity
≥99.0%
Solubility
DMSO 100 mg/mL (ultrasonic)
IRL 2500

IRL 2500

$356.50 USD