LE135

Vendor: Abmole

Type: Molecular

SKU: M13345

$207.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
LE135 is an effective RAR antagonist, which can selectively bind RARα (Ki is 1.4 μM) and RARβ (Ki is 220 nM), and has a higher affinity for RARβ. The LE135 is highly selective for RARγ, RXRα, RXRβ and RXRγ. LE135 is also a vitamin A acid receptor antagonist.
Casnumber
155877-83-1
Formula
C29H30N2O2
Mw
438.56
Psmiles
CC1(CCC(C2=CC3=C(C=C21)N=C(C4=CC=CC=C4N3C)C5=CC=C(C=C5)C(=O)O)(C)C)C
Purity
>99%
Solubility
DMSO ≥ 40 mg/mL
LE135

LE135

$207.00 USD