Loperamide hydrochloride

Vendor: Abmole

Type: Molecular

SKU: M2145

$63.25 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Loperamide hydrochloride is a high affinity μ-opioid receptor agonist with peripheral selectivity with Ki values of 2, 48 and 1156 nM for μ-, δ- and κ-opioid receptors respectively. Loperamide hydrochloride is also a selective and competitive human intestinal carboxylesterases (hiCE) inhibitor. It can be used to construct animal models of functional constipation.
Casnumber
34552-83-5
Formula
C29H33ClN2O2.HCl
Mw
513.51
Psmiles
Cl.CN(C)C(=O)C(CCN1CCC(O)(CC1)C2=CC=C(Cl)C=C2)(C3=CC=CC=C3)C4=CC=CC=C4
Purity
100.0%
Solubility
DMSO 30 mg/mL
Target synonyms
R-18553 hydrochloride
Loperamide hydrochloride

Loperamide hydrochloride

$63.25 USD