LP-935509

Vendor: Abmole

Type: Molecular

SKU: M28487

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$184.00 USD
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For research use only — not intended for clinical or diagnostic purposes.
LP-935509

LP-935509

$184.00 USD

THE SCIENCE, IN DETAIL

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Specifications
Bioactivity
LP-935509 is an orally active, potent, selective, ATP-competitive and brain-penetrant inhibitor of adaptor protein-2 associated kinase 1 (AAK1) with an IC50 of 3.3 nM and a Ki of 0.9 nM, respectively. LP-935509 is also a potent inhibitor of BIKE (IC50=14 nM) and a modest inhibitor of GAK (IC50=320 nM). LP-935509 shows antinociceptive activity. LP-935509 can be used for neuropathic pain and SARS-CoV-2 research.
Casnumber
1454555-29-3
Formula
C20H24N6O3
Mw
396.44
Psmiles
CC(C)OC(=O)N1CCN(CC1)C2=NC3=C(C=NN3C=C2)C4=C(N=CC=C4)OC
Purity
≥99.0%
Solubility
DMSO 50 mg/mL (ultrasonic)
Technical documents

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