Mavacamten (MYK-461)

Vendor: Abmole

Type: Molecular

SKU: M10262

$161.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Mavacamten, also known as SAR-439152 and MYK-461, is the first (first-class) orally bioavailable allosteric and reversible selective inhibitor of Cardiac Myosin. The IC50 of bovine heart and human heart was 490 nM and 711 nM, respectively.
Casnumber
1642288-47-8
Formula
C15H19N3O2
Mw
273.33
Psmiles
CC(C)N1C(=O)NC(=CC1=O)NC(C)C2=CC=CC=C2
Purity
99.80%
Solubility
DMSO 65 mg/mL
Target synonyms
SAR-439152; MYK-461
Mavacamten (MYK-461)

Mavacamten (MYK-461)

$161.00 USD