Mavatrep

Vendor: Abmole

Type: Molecular

SKU: M10841

$273.70 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Mavatrep is an orally active TRPV1 antagonist with high affinity for the hTRPV1 channel, inhibits the binding of the TRPV1 agonist to [3H]-Resiniferatoxin (Ki=6.5 nM), and has a low effect on the enzymatic activity of CYP subtypes 3A4, 1A2, and 2D6.
Casnumber
956274-94-5
Formula
C25H21F3N2O
Mw
422.45
Psmiles
CC(C)(C1=CC=CC=C1C2=CC3=C(C=C2)N=C(N3)C=CC4=CC=C(C=C4)C(F)(F)F)O
Purity
>99%
Solubility
DMSO ≥ 20 mg/mL
Target synonyms
JNJ-39439335
Mavatrep

Mavatrep

$273.70 USD