Meclinertant

Vendor: Abmole

Type: Molecular

SKU: M7330

$632.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Meclinertant (SR 48692) is an effective, selective, non-peptide and oral antagonist of active neurotensin receptor (NTS1). Meclinertant competitively antagonizes neurotensin-induced intracellular Ca2+ mobilization in human colon cancer cells, with a pA2 value of 8.13. Meclinertant has anti-anxiety, anti-addiction and memory disorder effects.
Casnumber
146362-70-1
Formula
C32H31ClN4O5
Mw
587.07
Psmiles
COC1=C(C(=CC=C1)OC)C2=CC(=NN2C3=C4C=CC(=CC4=NC=C3)Cl)C(=O)NC5(C6CC7CC(C6)CC5C7)C(=O)O
Purity
>98%
Solubility
DMSO 11.74 mg/mL
Target synonyms
SR 48692
Meclinertant

Meclinertant

$632.50 USD