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MK-8617

MK-8617

Regular price $862.50 USD
Sale price Regular price

THE SCIENCE, IN DETAIL

Know your product.

Specifications
Bioactivity
MK-8617 is an orally active pan-inhibitor of Hypoxia-inducible factor prolyl hydroxylase 1−3 (HIF PHD1−3), inhibiting PHD1, 2, 3 with IC50s of 1.0, 1.0 and 14 nM, respectively.
Casnumber
1187990-87-9
Formula
C24H21N5O4
Mw
443.45
Psmiles
COC1=CC=C(C=C1)C(NC(=O)C2=C(O)N=C(N=C2)C3=NN=CC=C3)C4=CC=C(OC)C=C4
Purity
>98.0%
Solubility
88 mg/mL in DMSO
Technical documents

Documents

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