Mozavaptan

Vendor: Abmole

Type: Molecular

SKU: M1917

$57.50 USD
Shipping calculated at checkout.

Documents

Coa

Available in stock (500)

  • Customs clearance fees may apply
  • Worldwide shipping available.
For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Mozavaptan (OPC-31260) is a benzazepine derivative and a potent, selective, competitive and orally active vasopressin V2 receptor antagonist with an IC50 of 14 nM. Mozavaptan shows ~85-fold selectivity for V2 receptor over V1 receptor (IC50 of 1.2 μM), and can antagonize the antidiuretic action of arginine vasopressin (AVP) in vivo.
Casnumber
137975-06-5
Formula
C27H29N3O2
Mw
427.53
Psmiles
CN(C)C1CCCN(C(=O)C2=CC=C(NC(=O)C3=C(C)C=CC=C3)C=C2)C4=C1C=CC=C4
Purity
99.12%
Solubility
DMSO 5 mg/mL
Target synonyms
OPC-31260
Mozavaptan

Mozavaptan

$57.50 USD