MS402

Vendor: Abmole

Type: Molecular

SKU: M10645

$138.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
MS402 is a novel BD1-selective BET BrD inhibitor, inhibiting primarily Th17 cell differentiation with a little or almost no effect on Th1 or Th2 and Treg cells. MS402 has Ki values of 77 nM, 718 nM, 110 nM, 200 nM, 83 nM, and 240 nM for BRD4(BD1), BRD4(BD2), BRD3(BD1), BRD3(BD2), BRD2(BD1) and BRD2(BD2), respectively.
Casnumber
1672684-68-2
Formula
C20H19ClN2O3
Mw
370.83
Psmiles
CC1=C(CCC1=O)NC2=C(C=C(C=C2)C(=O)NC3=CC=C(C=C3)OC)Cl
Purity
>98.5%
Solubility
DMSO ≥ 90 mg/mL
Target synonyms
MS-402
MS402

MS402

$138.00 USD