PCI-29732

Vendor: Abmole

Type: Molecular

SKU: M9889

$862.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
PCI-29732 is a potent, reversible BTK inhibitor with Kiapp values of 8.2, 4.6, and 2.5 nM for BTK, Lck, and Lyn, respectively, and has only modest inhibitory activity against Itk, another Tec family kinase. In addition, PCI 29732 inhibits the function of ABCG2 by competitively binding to the ATP binding site of ABCG2.
Casnumber
330786-25-9
Formula
C22H21N5O
Mw
371.44
Psmiles
NC1=NC=NC2=C1C(=N[N]2C3CCCC3)C4=CC=C(OC5=CC=CC=C5)C=C4
Purity
>99%
Solubility
DMSO ≥ 45 mg/mL
Target synonyms
PCI29732
PCI-29732

PCI-29732

$862.50 USD