PFI-2

Vendor: Abmole

Type: Molecular

SKU: M5128

$184.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
Casnumber
1627676-59-8
Formula
C23H25F4N3O3S
Mw
499.52
Psmiles
C1CCN(C1)C(=O)C(CC2=CC(=CC=C2)C(F)(F)F)NS(=O)(=O)C3=CC4=C(CNCC4)C(=C3)F
Purity
>98%
Solubility
DMSO 99 mg/mL; Water 4 mg/mL warmed
Target synonyms
(R)-PFI-2
PFI-2

PFI-2

$184.00 USD