Pico145

Vendor: Abmole

Type: Molecular

SKU: M14284

$322.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Pico145 (HC-608; Zerencotrep) is a remarkable inhibitor of TRPC1/4/5 channels, inhibits (−)-englerin A-activated TRPC4/TRPC5 channels, with IC50s of 0.349 and 1.3 nM in cells, and shows no effect on TRPC3, TRPC6, TRPV1, TRPV4, TRPA1, TRPM2, TRPM8.
Casnumber
1628287-16-0
Mw
524.88
Psmiles
CN1C2=C(C(=O)N(C1=O)CCCO)N(C(=N2)OC3=CC(=CC=C3)OC(F)(F)F)CC4=CC=C(C=C4)Cl
Purity
>99%
Solubility
DMSO ≥ 90 mg/mL
Target synonyms
HC-608; Zerencotrep
Pico145

Pico145

$322.00 USD