PU139

Vendor: Abmole

Type: Molecular

SKU: M28625

$281.75 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
PU139 is a potent pan-histone acetyltransferase (HAT) inhibitor. PU139 blocks the HATs Gcn5, p300/CBP-associated factor (PCAF), CREB (cAMP response element-binding) protein (CBP) and p300 with IC50s of 8.39, 9.74, 2.49 and 5.35 μM, respectively.
Casnumber
158093-65-3
Formula
C12H7FN2OS
Mw
246.26
Psmiles
C1=CC2=C(N=C1)SN(C2=O)C3=CC=C(C=C3)F
Purity
≥99.0%
Solubility
DMSO 10 mg/mL (ultrasonic and warming and heat to 60°C)
PU139

PU139

$281.75 USD