Pulrodemstat benzenesulfonate

Vendor: Abmole

Type: Molecular

SKU: M10727

$276.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
CC-90011 (Pulrodemstat) benzenesulfonate is a potent, selective, reversible and orally active lysine-specific demethylase-1 (LSD1) inhibitor,IC50 0.25 nM. CC-90011 benzenesulfonate has less enzymatic inhibition of LSD2, MOA-A and MAO-B. CC-90011 benzenesulfonate induces differentiation of acute myeloid leukemia (AML) and small cell lung cancer (SCLC) cells and has potent anti-cancer activity.
Casnumber
2097523-60-7
Formula
C30H29F2N5O5S
Mw
609.65
Psmiles
COC1=C(F)C=C(C=C1)C2=C(N=C(N(C)C2=O)N3CCC(N)CC3)C4=CC(=C(C=C4)C#N)F.O[S](=O)(=O)C5=CC=CC=C5
Purity
>99%
Solubility
DMSO ≥ 60 mg/mL
Target synonyms
CC-90011 benzenesulfonate
Pulrodemstat benzenesulfonate

Pulrodemstat benzenesulfonate

$276.00 USD