R406 besylate

Vendor: Abmole

Type: Molecular

SKU: M14916

$224.25 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
R406 is an orally available and competitive Syk/FLT3 inhibitor for ATP binding with a Ki of 30 nM, potently inhibits Syk kinase activity in vitro with an IC50 of 41 nM, measured at an ATP concentration corresponding to its Km value.
Casnumber
841290-81-1
Formula
C22H23FN6O5.C6H6O3S
Mw
628.63
Psmiles
COC1=C(OC)C(=CC(=C1)NC2=NC(=C(F)C=N2)NC3=NC4=C(OC(C)(C)C(=O)N4)C=C3)OC.O[S](=O)(=O)C5=CC=CC=C5
Purity
>98.5%
Solubility
DMSO ≥ 61 mg/mL
Target synonyms
R406 benzenesulfonate; Tamatinib
R406 besylate

R406 besylate

$224.25 USD