Relacorilant

Vendor: Abmole

Type: Molecular

SKU: M11555

$511.75 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Relacorilant is a selective, oral bioeffective glucocorticoid receptor antagonist (Ki of 7.2 nM in HepG2 TAT assay and 12,81.2 nM in rat, human and monkey glucocorticoid receptor in cell-based assay). Relacorilant can be used in studies of Cushing's syndrome.
Casnumber
1496510-51-0
Formula
C27H22F4N6O3S
Mw
586.56
Psmiles
C[N]1C=C(C=N1)[S;v6](=O)(=O)N2CCC3=CC4=C(CC3(C2)C(=O)C5=CC(=CC=N5)C(F)(F)F)C=N[N]4C6=CC=C(F)C=C6
Purity
99.50%
Solubility
DMSO ≥ 60 mg/mL
Target synonyms
CORT 125134
Relacorilant

Relacorilant

$511.75 USD