RSM-932A

Vendor: Abmole

Type: Molecular

SKU: M30694

$1,437.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
RSM-932A (TCD-717) is a specific ChoKα inhibitor with IC50s of 1 and 33 μM for human recombinant ChoKα and ChoKβ enzymes, respectively. RSM-932A acts as the “first in humans” compound targeting ChoKα. RSM-932A is potent in vitro anti-proliferative and in vivo anti-tumoral activity against human xenografts in mice, showing high efficacy with low toxicity profiles.
Casnumber
850807-63-5
Formula
C46H38Br2Cl2N4
Mw
877.53
Psmiles
CN(C1=CC=C(C=C1)Cl)C2=CC=[N+](C3=CC=CC=C32)CC4=CC=C(C=C4)C5=CC=C(C=C5)C[N+]6=CC=C(C7=CC=CC=C76)N(C)C8=CC=C(C=C8)Cl.[Br-].[Br-]
Purity
≥99.0%
Solubility
DMSO 16.67 mg/mL (ultrasonic and warming and heat to 60°C)
Target synonyms
TCD-717
RSM-932A

RSM-932A

$1,437.50 USD