Apatinib (YN968D1) mesylate

Name: Apatinib (YN968D1) mesylate
Brand: Selleckchem
Price: 240.0 USD
Availability: InStock

Vendor: Selleckchem

Type: Protein Tyrosine Kinase

SKU: S2221-10mg

$240.00 USD

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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Big target

Protein Tyrosine Kinase

Cas number

1218779-75-9

Formula

C25H27N5O4S

Small target

VEGFR

Smiles

C[S](O)(=O)=O.O=C(NC1=CC=C(C=C1)C2(CCCC2)C#N)C3=CC=CN=C3NCC4=CC=NC=C4

Storage conditions

2 years -80 in solvent

Synonyms

YN968D1, Rivoceranib

Background

Apatinib mesylate (YN968D1, Rivoceranib) is a potent inhibitor of the VEGF signaling pathway with IC50 values of 1 nM, 13 nM, 429 nM and 530 nM for VEGFR-2, Ret (c-Ret), c-Kit and c-Src, respectively. Apatinib mesylate induces both autophagy and apoptosis.

Apatinib (YN968D1) mesylate

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Product Overview

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