GSK256066 chemical structure

GSK256066

Vendor: Selleckchem

Type: Metabolism

SKU: S2620-10mg

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$278.00 USD
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For research use only — not intended for clinical or diagnostic purposes.
GSK256066 chemical structure

GSK256066

$278.00 USD

THE SCIENCE, IN DETAIL

Know your product.

Specifications
Big target
Metabolism
Cas number
801312-28-7
Formula
C27H26N4O5S
Small target
PDE
Smiles
CC1=CC(=CC2=C(C(=CN=C12)C(=O)N)NC3=CC(=CC=C3)OC)S(=O)(=O)C4=CC=CC(=C4)C(=O)N(C)C
Storage conditions
2 years -80 in solvent
Scientific background
GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.Phase 2.
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